Last update 20 Mar 2025

SMARCA2 inhibitors (Arvinas LLC)

Overview

Basic Info

Drug Type
Proteolysis-targeting chimeras (PROTAC)
Synonyms-
Target
SMARCA2
Action
inhibitors
Mechanism
SMARCA2 inhibitors(Probable global transcription activator SNF2L2 inhibitors)
Therapeutic Areas
Neoplasms
Active Indication
Neoplasms
Inactive Indication-
Originator Organization-
Active Organization
Arvinas Operations, Inc.Genentech, Inc.Genentech, Inc.
Inactive Organization-
Drug Highest PhasePreclinical
First Approval Date-
Regulation-

Related

100 Clinical Results associated with SMARCA2 inhibitors (Arvinas LLC)
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100 Translational Medicine associated with SMARCA2 inhibitors (Arvinas LLC)
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100 Patents (Medical) associated with SMARCA2 inhibitors (Arvinas LLC)
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1
Literatures (Medical) associated with SMARCA2 inhibitors (Arvinas LLC)
25 Jan 2024Journal of Medicinal ChemistryQ1 · MEDICINE
PROTACs Targeting BRM (SMARCA2) Afford Selective In Vivo Degradation over BRG1 (SMARCA4) and Are Active in BRG1 Mutant Xenograft Tumor Models
Q1 · MEDICINE
100 Deals associated with SMARCA2 inhibitors (Arvinas LLC)
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R&D Status

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IndicationHighest PhaseCountry/LocationOrganizationDate
NeoplasmsPreclinical
United States
Genentech, Inc.Genentech, Inc.
05 Jan 2024
NeoplasmsPreclinical
United States
Arvinas Operations, Inc.
05 Jan 2024
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Clinical Result

Indication
Phase
Evaluation
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Phase
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Deal

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Approval

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Regulation

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