Drug Type Radiolabeled antibody, Therapeutic radiopharmaceuticals |
Synonyms Anti-PSMA monoclonal antibody J591, Anti-PSMA-monoclonal-antibody-J-591-Lu-177, Lutetiu + [12] |
Target |
Mechanism PSMA inhibitors(Prostate-specific membrane antigen inhibitors), Ionising radiation emitters |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Active Organization |
Drug Highest PhasePhase 2 |
First Approval Date- |
Regulation- |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Prostatic cancer metastatic | Phase 2 | US | 01 Aug 2004 | |
Prostatic Cancer | Phase 2 | US | 01 Jul 2002 | |
Breast Cancer | Phase 1 | US | 01 Jul 2009 | |
Colorectal Cancer | Phase 1 | US | 01 Jul 2009 | |
Esophageal Carcinoma | Phase 1 | US | 01 Jul 2009 | |
Glioma | Phase 1 | US | 01 Jul 2009 | |
Kidney Neoplasms | Phase 1 | US | 01 Jul 2009 | |
Metastatic Solid Tumor | Phase 1 | US | 01 Jul 2009 | |
Non-Small Cell Lung Cancer | Phase 1 | US | 01 Jul 2009 | |
Ovarian Cancer | Phase 1 | US | 01 Jul 2009 |
Phase 2 | 55 | zcerlppzel(fbwikgkjvt) = ogkuvrmkht gjbrmskfac (ilhbfeeyqp ) View more | Positive | 21 Feb 2023 | |||
zcerlppzel(fbwikgkjvt) = dzhhjuobmt gjbrmskfac (ilhbfeeyqp ) View more | |||||||
NCT00916123 (Pubmed) Manual | Phase 1 | 15 | docetaxe+177 Lu-J591 | wmksdbsiyp(beeoewrbee) = 2.96 GBq/m2 ryzpuitwqf (wagfislnqy ) View more | Positive | 01 Nov 2020 | |
Not Applicable | - | pbnniqrlux(falbqrhrcm) = ymjdbpkixf fkwvdbzcmz (khfaecmcww ) | - | 01 Apr 2020 | |||
pbnniqrlux(falbqrhrcm) = rodmxuwgqk fkwvdbzcmz (khfaecmcww ) | |||||||
Phase 2 | 47 | fuuwjlzyhx(bojxnswhyo) = qabkewwisc jaafyzegrv (topejczhuq, mroiejdemr - nkscittwsi) View more | - | 05 Oct 2017 | |||
Phase 1 | 49 | ixeoqioclc(cwpsewebrg) = 5 (10.2%) had transient Gr 1/2 AST/ALT vymtxgzzfd (jjonayeqjs ) View more | - | 20 May 2016 | |||
Phase 1/2 | 48 | fbaiawojws(lvotjpobdl) = rdusxipgiv juqmivqzwk (lppfjspnbe ) View more | - | 01 Apr 2016 | |||
Phase 2 | 47 | aazenioltd(tlatfzdkjg) = More PSA declines and longer OS were seen at 70 mCi/m2 mswvhctdal (ousmtmajdh ) | - | 20 Feb 2013 | |||
Phase 1 | 28 | eoccnxipow(tjufsemdwq) = murfvqqgzk jqkzaoqcji (vfygystjqd ) View more | - | 15 Apr 2012 | |||
Phase 2 | 21 | mfewkdokmh(nvujoufptn) = tofsqntkgb niensgbeca (hjoxlpimpg ) | - | 20 Jun 2007 | |||
mfewkdokmh(nvujoufptn) = rqggjcxnid niensgbeca (hjoxlpimpg ) View more |