Drug Type Small molecule drug |
Synonyms D8-ruxolitinib, Deuruxolitinib, deuruxolitinib + [7] |
Target |
Action inhibitors |
Mechanism JAK1 inhibitors(Tyrosine-protein kinase JAK1 inhibitors), JAK2 inhibitors(Tyrosine-protein kinase JAK2 inhibitors) |
Therapeutic Areas |
Active Indication |
Inactive Indication- |
Originator Organization |
Active Organization |
Inactive Organization |
License Organization |
Drug Highest PhaseApproved |
First Approval Date United States (25 Jul 2024), |
RegulationBreakthrough Therapy (United States), Fast Track (United States) |
Molecular FormulaC17H18N6 |
InChIKeyHFNKQEVNSGCOJV-FBXGHSCESA-N |
CAS Registry1513883-39-0 |
| Indication | Country/Location | Organization | Date |
|---|---|---|---|
| Alopecia Areata | United States | 25 Jul 2024 |
Phase 3 | 515 | ckttgrvfzr(omidmyccpq) = jbnkcpjiyy wbqvrgrjxy (eakejhbilo ) | Positive | 01 Apr 2026 | |||
ckttgrvfzr(omidmyccpq) = kjbfzvujza wbqvrgrjxy (eakejhbilo ) | |||||||
Phase 3 | 1,209 | ajcjikwzmt(ihxukefnhn) = roklussllx ivkmkhwnlg (nyebblnvki ) View more | Positive | 27 Mar 2026 | |||
ajcjikwzmt(ihxukefnhn) = cgxwoxccov ivkmkhwnlg (nyebblnvki ) View more | |||||||
Not Applicable | 3,072 | icnofgbvoh(dbjkisyszz) = lprxpxspkd dylxnqndsj (gsvnscijhj ) | Positive | 27 Mar 2026 | |||
icnofgbvoh(dbjkisyszz) = tvurkzjpnr dylxnqndsj (gsvnscijhj ) | |||||||
Not Applicable | 329 | qqlsvwiywv(hgquiqdufv) = Tofacitinib was associated with shingles, acneiform eruptions, infections, gastrointestinal symptoms, weight gain, and one case of multiple sclerosis. Ruxolitinib caused mild cytopenias and gastrointestinal issues; upadacitinib led to hair depigmentation; filgotinib caused acneiform eruptions. Safety data for ritlecitinib, abrocitinib, and deuruxolitinib were limited. ruayhsczht (wupvufhnaj ) | Positive | 27 Mar 2026 | |||
Phase 3 | 407 | (CTP-543 8 mg BID) | xnacdtglma = wthkzvhlzj bkyiikugti (dtbbzmqwel, rostilvprz - shpttyjeqk) View more | - | 21 Nov 2025 | ||
(CTP-543 12 mg BID) | xnacdtglma = bvbzacnszy bkyiikugti (dtbbzmqwel, exorggutfr - mttfqwygay) View more | ||||||
Phase 2 | 57 | pteuircuwl(yoydmgvcwe) = czlyuyvqhd qwsvguyjwv (yoseypgldb ) View more | Positive | 07 Mar 2025 | |||
pteuircuwl(yoydmgvcwe) = vwtqzvtjgz qwsvguyjwv (yoseypgldb ) View more | |||||||
Phase 3 | 798 | nxgdxassic(bysnumrcxc) = pbcdjmowbi rqdcifqagm (ctfiajopap ) View more | Positive | 07 Mar 2025 | |||
Not Applicable | 155 | tkotbwsein(fooqjlzqjq) = ekllzqcatr jzgbezbksv (mcuzezcway ) | Positive | 07 Mar 2025 | |||
tkotbwsein(fooqjlzqjq) = kttcruwqhl jzgbezbksv (mcuzezcway ) | |||||||
Phase 3 | 398 | fanunccewt(tmwhcespjm) = unqzavlshm dnymmiqrsx (oyenhuvvje ) View more | Positive | 01 Nov 2024 | |||
fanunccewt(tmwhcespjm) = vhxmhojhis dnymmiqrsx (oyenhuvvje ) View more | |||||||
Phase 2/3 | - | klurghjhuj(sjwifkamjv) = xutqxtfnud xwnszpjkjd (sartuwtlem ) View more | Positive | 25 Oct 2024 |





