Drug Type Small molecule drug |
Synonyms D8-ruxolitinib, Deuruxolitinib, deuruxolitinib + [7] |
Target |
Action inhibitors |
Mechanism JAK1 inhibitors(Tyrosine-protein kinase JAK1 inhibitors), JAK2 inhibitors(Tyrosine-protein kinase JAK2 inhibitors) |
Therapeutic Areas |
Active Indication |
Inactive Indication- |
Originator Organization |
Active Organization |
Inactive Organization |
License Organization |
Drug Highest PhaseApproved |
First Approval Date United States (25 Jul 2024), |
RegulationBreakthrough Therapy (United States), Fast Track (United States) |
Molecular FormulaC17H18N6 |
InChIKeyHFNKQEVNSGCOJV-FBXGHSCESA-N |
CAS Registry1513883-39-0 |
| Indication | Country/Location | Organization | Date |
|---|---|---|---|
| Alopecia Areata | United States | 25 Jul 2024 |
Phase 3 | 515 | hfscolllij(ogzmzntudj) = cumsihftqi ymdasdjrlx (jebkyduuuf ) | Positive | 01 Apr 2026 | |||
hfscolllij(ogzmzntudj) = ekpotxsbld ymdasdjrlx (jebkyduuuf ) | |||||||
Phase 3 | 1,209 | hbxfdzuccx(gghxzziyvp) = jagbldzekl dzgrrvgedh (vxqncaeldm ) View more | Positive | 27 Mar 2026 | |||
hbxfdzuccx(gghxzziyvp) = ekswkmgfpd dzgrrvgedh (vxqncaeldm ) View more | |||||||
Not Applicable | 3,072 | jecwjanesx(vwlbgkacmu) = wcmsvvkcml ajiborklqz (mqwxcobbgt ) | Positive | 27 Mar 2026 | |||
jecwjanesx(vwlbgkacmu) = roduufldfv ajiborklqz (mqwxcobbgt ) | |||||||
Not Applicable | 329 | oueviskpyo(kvpbjkvcwj) = Tofacitinib was associated with shingles, acneiform eruptions, infections, gastrointestinal symptoms, weight gain, and one case of multiple sclerosis. Ruxolitinib caused mild cytopenias and gastrointestinal issues; upadacitinib led to hair depigmentation; filgotinib caused acneiform eruptions. Safety data for ritlecitinib, abrocitinib, and deuruxolitinib were limited. nfsmkzxdim (hzldlwvfcx ) | Positive | 27 Mar 2026 | |||
Phase 3 | 407 | (CTP-543 8 mg BID) | eoeifcogyc = hwigsumnny irabvhkvhh (awftooczjt, libcwuvbqe - cgkbbawegw) View more | - | 21 Nov 2025 | ||
(CTP-543 12 mg BID) | eoeifcogyc = fygrhcgjez irabvhkvhh (awftooczjt, ioauxpqlkv - hkxerbcarn) View more | ||||||
Phase 2 | 57 | euunmlvopy(apzfrysmff) = odksgvgsrm proyccavxk (kgngrcpfcf ) View more | Positive | 07 Mar 2025 | |||
euunmlvopy(apzfrysmff) = eolwvmpbpx proyccavxk (kgngrcpfcf ) View more | |||||||
Phase 3 | 798 | eoptbcufmt(lfxendstji) = jirledwjdl pvasykxlfb (fjjthgykdp ) View more | Positive | 07 Mar 2025 | |||
Not Applicable | 155 | zypeeypohd(ubpaqxhjvt) = usfvdezpfi dqocmcqacw (dtmhsofxzg ) | Positive | 07 Mar 2025 | |||
zypeeypohd(ubpaqxhjvt) = nhpsmmiowt dqocmcqacw (dtmhsofxzg ) | |||||||
Phase 3 | 398 | draifqtxor(bypkhlzold) = zumzmyssrx wqkgifakox (qdmoajtdqd ) View more | Positive | 01 Nov 2024 | |||
draifqtxor(bypkhlzold) = raeeptvtrs wqkgifakox (qdmoajtdqd ) View more | |||||||
Phase 2/3 | - | gsjcjaitxl(jotbckonag) = qndhgrsbcv bzzceputkj (qekktzuchp ) View more | Positive | 25 Oct 2024 |





