Last update 19 Apr 2025

Gamcemetinib

Overview

Basic Info

Drug Type
Small molecule drug
Synonyms
BMS 986371, BMS-986371, BMS986371
+ [2]
Target
Action
inhibitors
Mechanism
MAPKAPK2 inhibitors(MAP kinase-activated protein kinase 2 inhibitors)
Active Indication-
Originator Organization
Active Organization-
Drug Highest PhaseDiscontinuedPhase 2
First Approval Date-
Regulation-
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Structure/Sequence

Molecular FormulaC22H20ClN5O3S
InChIKeyPYOQIOLRFIRRSO-LLVKDONJSA-N
CAS Registry1887069-10-4

R&D Status

10 top R&D records.
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IndicationHighest PhaseCountry/LocationOrganizationDate
Ankylosing SpondylitisPhase 2
United States
25 Aug 2021
Ankylosing SpondylitisPhase 2
Czechia
25 Aug 2021
Ankylosing SpondylitisPhase 2
Germany
25 Aug 2021
Ankylosing SpondylitisPhase 2
Poland
25 Aug 2021
Ankylosing SpondylitisPhase 2
Romania
25 Aug 2021
Ankylosing SpondylitisPhase 2
Spain
25 Aug 2021
Ankylosing SpondylitisPhase 2
Turkey
25 Aug 2021
InflammationPhase 1
United Kingdom
23 May 2018
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Clinical Result

Indication
Phase
Evaluation
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Study
Phase
PopulationAnalyzed EnrollmentGroupResultsEvaluationPublication Date
Phase 2
167
Placebo
(Placebo Biologic Naive)
gdkvnoxkoo = toarondmwu lavsoxgsno (qcjrmkyezu, iotawvwuok - zfnftzkufr)
-
01 May 2024
(CC-99677 60 mg Biologic Naive)
gdkvnoxkoo = iibbbcidic lavsoxgsno (qcjrmkyezu, swcdvtpujv - vfclxvoums)
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Deal

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Core Patent

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Clinical Trial

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Approval

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Regulation

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