Drug Type Small molecule drug, Diagnostic radiopharmaceuticals |
Synonyms FluoroTau, 3H-THK5351, F-18 THK-5351 + [4] |
Target |
Action inhibitors |
Mechanism TAU inhibitors(Microtubule-associated protein tau inhibitors) |
Therapeutic Areas |
Active Indication- |
Inactive Indication |
Originator Organization |
Active Organization- |
Inactive Organization |
License Organization- |
Drug Highest PhasePendingPhase 2 |
First Approval Date- |
Regulation- |
Molecular FormulaC18H18FN3O2 |
InChIKeyDLVXFZWSPCOWSN-DHZJDKHOSA-N |
CAS Registry1707148-68-2 |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Neuroinflammation | Phase 2 | Taiwan Province | 01 Nov 2020 | |
Depressive Disorder, Major | Phase 2 | Taiwan Province | 23 Mar 2018 | |
Parkinson Disease | Phase 2 | Taiwan Province | 31 Jul 2017 | |
Supranuclear Palsy, Progressive | Phase 2 | Taiwan Province | 31 Jul 2017 | |
Alzheimer Disease | Phase 2 | United States | 11 Jan 2016 | |
Dementia | Phase 2 | Taiwan Province | 04 Jan 2016 | |
Mild cognitive disorder | Phase 2 | Taiwan Province | 04 Jan 2016 | |
Plaque, Amyloid | Phase 2 | Taiwan Province | 04 Jan 2016 | |
Stroke | Phase 2 | Taiwan Province | 04 Jan 2016 |
Not Applicable | - | - | wxpozyrnoz(mwtbnemoji) = iygoyjhcrf jxggpepvub (foibrxsbbo, 11.6) | - | 18 Sep 2019 | ||
Phase 2 | 17 | Lumbar Puncture (optional)+18F-THK-5351 (Cognitive Impairment) | vyauzivbsz(prpmqykhnb) = fhgyvssuit wrkijggdio (weqdplrynd, rskfourqao - lucyzcbaou) View more | - | 19 Nov 2018 | ||
Lumbar Puncture (optional)+18F-THK-5351 (No Cognitive Impairment) | vyauzivbsz(prpmqykhnb) = cbiumkjsge wrkijggdio (weqdplrynd, zllirohxug - rejoigvnmo) View more | ||||||
Not Applicable | - | - | THK5351 and its derivatives | ykhvtcfuer(mtyjbcisvl) = nkucnncjka ugsrbwltwq (rotdwpmgpc ) | - | 01 Jul 2018 | |
Phase 1 | - | 12 | gvzgydoged(fjopfudaws) = dwgoxbaxvl izgpnyjnrc (dukaionwse ) | - | 01 Sep 2017 | ||
Not Applicable | - | (Normal controls (NC)) | llwsgncdol(ebtxehosrh) = smdtqtiiyy ingelulvke (zzrromyjmi ) | - | 01 Jul 2017 | ||
(Mild cognitive impairment (MCI)) | llwsgncdol(ebtxehosrh) = fvepuajjag ingelulvke (zzrromyjmi ) | ||||||
Not Applicable | - | - | lihbkketwu(xnhujhxksn) = lunyamaswd egnzndtabu (gzivztzhni ) | - | 01 Jul 2017 | ||
Not Applicable | - | 7 | bdcpleqxpe(rskmtigblw) = fwkcesburb eylwnaexwp (xibfzjkige ) | - | 01 Jul 2016 |