Drug Type Small molecule drug, Diagnostic radiopharmaceuticals |
Synonyms FluoroTau, 3H-THK5351, F-18 THK-5351 + [4] |
Target |
Action inhibitors |
Mechanism TAU inhibitors(Microtubule-associated protein tau inhibitors) |
Therapeutic Areas |
Active Indication- |
Inactive Indication |
Originator Organization |
Active Organization- |
Inactive Organization |
License Organization- |
Drug Highest PhasePendingPhase 2 |
First Approval Date- |
Regulation- |
Molecular FormulaC18H18FN3O2 |
InChIKeyDLVXFZWSPCOWSN-DHZJDKHOSA-N |
CAS Registry1707148-68-2 |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Neuroinflammation | Phase 2 | Taiwan Province | 01 Nov 2020 | |
Depressive Disorder, Major | Phase 2 | Taiwan Province | 23 Mar 2018 | |
Parkinson Disease | Phase 2 | Taiwan Province | 31 Jul 2017 | |
Supranuclear Palsy, Progressive | Phase 2 | Taiwan Province | 31 Jul 2017 | |
Alzheimer Disease | Phase 2 | United States | 11 Jan 2016 | |
Dementia | Phase 2 | Taiwan Province | 04 Jan 2016 | |
Mild cognitive disorder | Phase 2 | Taiwan Province | 04 Jan 2016 | |
Plaque, Amyloid | Phase 2 | Taiwan Province | 04 Jan 2016 | |
Stroke | Phase 2 | Taiwan Province | 04 Jan 2016 |
Not Applicable | - | - | kxbklndlmb(ccrggjljzj) = kybfydqdak nufonubayl (ajvinfaxwz, 11.6) | - | 18 Sep 2019 | ||
Phase 2 | 17 | Lumbar Puncture (optional)+18F-THK-5351 (Cognitive Impairment) | bjbumwbvlf(azmgyqxktq) = dfpnccaqvl zunptqvrhq (fgyylgtcrc, thpvkoodgy - otmpplzxyy) View more | - | 19 Nov 2018 | ||
Lumbar Puncture (optional)+18F-THK-5351 (No Cognitive Impairment) | bjbumwbvlf(azmgyqxktq) = yqxcvalbvl zunptqvrhq (fgyylgtcrc, jerrnzgzya - kvqqhzmmex) View more | ||||||
Not Applicable | - | - | THK5351 and its derivatives | bxwurkjgxc(qboyhbopga) = hzezkilzbv noqovwnsrl (bwppgtdtuj ) | - | 01 Jul 2018 | |
Phase 1 | - | 12 | ximptrtjro(dlzdhrdbnu) = szglavkbkh trprjkmvta (ryqzogabgq ) | - | 01 Sep 2017 | ||
Not Applicable | - | (Normal controls (NC)) | mvngzcdrxo(etmvgvdbod) = faqerqalst hdbukgldaq (epfiyeowyh ) | - | 01 Jul 2017 | ||
(Mild cognitive impairment (MCI)) | mvngzcdrxo(etmvgvdbod) = wdkayzqvfd hdbukgldaq (epfiyeowyh ) | ||||||
Not Applicable | - | - | otbuqdydxa(eqsreyijnw) = qkpiaoowej ielouadsrf (gxvofbwygv ) | - | 01 Jul 2017 | ||
Not Applicable | tau protein | - | nhqxwofoxa(xxdhijptki) = hwludlhwus mzeacwzzbf (gaeryjskyw ) View more | - | 21 Sep 2016 | ||
Not Applicable | - | 7 | prqzwdvonb(ztgsljmkga) = qoktivngdc xlrvvatkhs (yhuuaznmrc ) | - | 01 Jul 2016 |