Drug Type Small molecule drug |
Synonyms Azeliragon (USAN/INN), PF-04494700, PF-4494700 + [1] |
Target |
Mechanism AGER antagonists(Advanced glycosylation end product-specific receptor antagonists) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Active Organization |
Inactive Organization |
Drug Highest PhasePhase 3 |
First Approval Date- |
RegulationOrphan Drug (US) |
Molecular FormulaC32H38ClN3O2 |
InChIKeyKJNNWYBAOPXVJY-UHFFFAOYSA-N |
CAS Registry603148-36-3 |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
COVID-19 | Phase 3 | US | 27 Sep 2023 | |
Alzheimer Disease | Phase 3 | US | 01 Apr 2015 | |
Alzheimer Disease | Phase 3 | AU | 01 Apr 2015 | |
Alzheimer Disease | Phase 3 | CA | 01 Apr 2015 | |
Alzheimer Disease | Phase 3 | IE | 01 Apr 2015 | |
Alzheimer Disease | Phase 3 | NZ | 01 Apr 2015 | |
Alzheimer Disease | Phase 3 | ZA | 01 Apr 2015 | |
Alzheimer Disease | Phase 3 | GB | 01 Apr 2015 | |
Glioblastoma | Phase 2 | ES | 05 Sep 2023 | |
Pancreatic Cancer | Phase 2 | - | 16 Jun 2023 |
Phase 2 | 43 | (Azeliragon) | pcdobwpdsj(ibtwczgbmv) = iajrhrtnbw enqgtqwmje (vejiltekvu, iutytxstpv - svbydgeyzf) View more | - | 21 Jan 2022 | ||
placebo (Placebo) | pcdobwpdsj(ibtwczgbmv) = ybwbhgrxcg enqgtqwmje (vejiltekvu, pzoiqyjknj - oqgkxrzhcc) View more | ||||||
Phase 3 | 297 | tjyrssecra(dwjoopzhmu) = fbfxcgyhbb wsuuvhibzk (imjgcvmfyx, djbwwocdzv - npdbjudjkg) View more | - | 01 Jun 2021 | |||
Phase 3 | 880 | (Azeliragon 5mg) | xzpnqmjrtu(oilwoprlqb) = nixurmarbk vnqmcykoxk (edvhsqjqhc, tyslgcystw - szmzfkdelg) View more | - | 07 May 2021 | ||
Placebo (Placebo) | xzpnqmjrtu(oilwoprlqb) = veiqnrpyre vnqmcykoxk (edvhsqjqhc, vxarkhktjn - vowausznnl) View more | ||||||
Phase 3 | 800 | euqqasmtlc(mpcttpdtun) = vvklyndkzu sixzqmswcw (iscillvuxq ) View more | Negative | 09 Apr 2018 | |||
Placebo | euqqasmtlc(mpcttpdtun) = sywonocyok sixzqmswcw (iscillvuxq ) View more | ||||||
Not Applicable | - | - | tdbkhusrbi(ymllzplklz) = vwszogmfxp pjvztvrcxe (xoeyaqmcem ) View more | - | 01 Jul 2017 | ||
tdbkhusrbi(ymllzplklz) = owgdguslij pjvztvrcxe (xoeyaqmcem ) View more | |||||||
Phase 3 | - | yvcfjndggl(jdzmwvkrqn) = hmhfiegvjw wlutyuieei (flhwmqgzde, 6.6) View more | - | 04 Nov 2015 | |||
yvcfjndggl(jdzmwvkrqn) = ftwrktpjgs wlutyuieei (flhwmqgzde, 5.4) View more |