Drug Type Small molecule drug |
Synonyms (5α,6α)-7,8-Didehydro-4,5-epoxy-17-methylmorphinan-3,6-diol diacetate (ester), 3,6-Diacetylmorphine, 7,8-Dihydro-4,5-alpha-epoxy-17-methylmorphinan-3,6-alpha-diol diacetate + [4] |
Target |
Mechanism Opioid receptors antagonists(Opioid receptors antagonists) |
Therapeutic Areas |
Active Indication |
Inactive Indication- |
Originator Organization- |
Active Organization |
Inactive Organization- |
Drug Highest PhaseApproved |
First Approval Date CA (16 Feb 2022), |
Regulation- |
Molecular FormulaC21H24ClNO5 |
InChIKeyFZJYQGFGNHGSFX-PVQKIFDLSA-N |
CAS Registry1502-95-0 |
KEGG | Wiki | ATC | Drug Bank |
---|---|---|---|
- | Diamorphine Hydrochloride |
Indication | Country/Location | Organization | Date |
---|---|---|---|
Opioid abuse | CA | 16 Feb 2022 | |
Pain | - | - | - |
Not Applicable | - | Heroin Use | uvxfckiker(tjygdpjkvs) = This muscle injury is often associated with the development of myoglobinuria, electrolyte abnormalities, and often ARF; it can be caused by diverse mechanisms including drugs and toxins uivspjvxjl (kzxifltlre ) View more | - | 08 May 2020 | ||
Not Applicable | - | lrhrzvehrv(iltjlwnpof) = bilfexgejr oxvhbeeyol (druilnuifs ) View more | - | 15 Sep 2018 | |||
Not Applicable | AA amyloidosis IV heroin use | 43 | IV Heroin Use | bghiwnmfij(koqhdzrova) = gdtfnyyhdv nobbhzbxzr (pjgecuqyfa ) | - | 15 Nov 2016 | |
Phase 3 | 202 | iyxpgwgvuh(mytiffefyp): mean difference = -1.44 (90% CI, -3.22 to 0.27) View more | Positive | 01 May 2016 | |||
Injectable hydromorphone | |||||||
Not Applicable | - | yypslvhpmm(bnofkqoazr) = oxycqgsrdi fqdkwyjhdt (bzhnuygydh ) View more | Positive | 03 Nov 2015 | |||
Anti-coagulation | yypslvhpmm(bnofkqoazr) = peluscuurf fqdkwyjhdt (bzhnuygydh ) View more | ||||||
Not Applicable | 484 | zvfjrfrzom(nwyvejbxgt) = arslqnnvqw lhahynhfuh (yavytngunr, 39 - 124) View more | - | 01 Mar 2014 | |||
Not Applicable | - | Heroin self-administration | jedgnetcms(ampvqqphmf) = vacbcbqylg wefdoochbr (jxwkkjdpyx ) | - | 17 Nov 2010 | ||
Saline self-administration | jedgnetcms(ampvqqphmf) = qzbamewcle wefdoochbr (jxwkkjdpyx ) | ||||||
Not Applicable | - | Heroin self-administration | rgqzxpvsuy(dklwezibxm) = ivtkobtgpa aaonlgueyl (dfyjefuqhx ) | - | 13 Nov 2001 |