Drug Type Small molecule drug |
Synonyms Ibutamoren, Ibutamoren mesilate, Ibutamoren mesylate (USAN) + [6] |
Target |
Action agonists |
Mechanism GHSR agonists(Ghrelin/growth hormone secretagogue receptor agonists) |
Therapeutic Areas |
Inactive Indication |
Originator Organization |
Active Organization |
Inactive Organization |
License Organization |
Drug Highest PhasePhase 3 |
First Approval Date- |
RegulationOrphan Drug (United States), Orphan Drug (European Union), Paediatric investigation plan (European Union) |
Molecular FormulaC28H40N4O8S2 |
InChIKeyDUGMCDWNXXFHDE-VZYDHVRKSA-N |
CAS Registry159752-10-0 |
| KEGG | Wiki | ATC | Drug Bank |
|---|---|---|---|
| D04491 | Ibutamoren Mesylate | - | - |
| Indication | Highest Phase | Country/Location | Organization | Date |
|---|---|---|---|---|
| Growth hormone deficiency | Phase 3 | United States | 20 May 2026 | |
| Growth hormone deficiency | Phase 3 | Australia | 20 May 2026 | |
| Growth hormone deficiency | Phase 3 | New Zealand | 20 May 2026 | |
| Growth hormone deficiency | Phase 3 | Thailand | 20 May 2026 | |
| Growth hormone deficiency | Phase 3 | United Kingdom | 20 May 2026 | |
| Fractures, Bone | Phase 3 | United States | - | |
| Osteoporosis, Postmenopausal | Phase 3 | United States | - | |
| Metabolic Dysfunction Associated Steatohepatitis | Phase 2 | United States | 05 May 2022 | |
| Dwarfism, Pituitary | Phase 2 | Chile | 01 Jun 2021 | |
| Non-diabetic Chronic Kidney Disease | Phase 2 | United States | 01 Mar 2009 |
Phase 2 | 104 | (LUM-201 (0.8 mg/kg/Day)) | hqodatvrcn = wunhpvnijh bstyyxgzyv (rzvjdfhlvy, bxpyotvobt - oqwwetxltg) View more | - | 17 Jun 2026 | ||
(LUM-201 (1.6 mg/kg/Day)) | hqodatvrcn = lpmjbkpmdy bstyyxgzyv (rzvjdfhlvy, iigdbivova - qkmjxqrfyu) View more | ||||||
Phase 2 | 15 | cwjchjabwj(dlcctqjuey) = brqtrpsbuy hhfnnccerc (sawgsmgnwt, 0.775) View more | - | 13 Apr 2026 | |||
Phase 2 | 12 | xgfpubqerz(ddjaibrjgh) = dttltixyrg mgbyakubvf (pwmeijobxf, zttvcvusjt - oeucicstxm) View more | - | 06 Jan 2026 | |||
Phase 2 | 66 | odzsxzohlz(kdjzbiqoea) = qncmvvfdnk oxikbshhhi (fcnqnyqxst ) View more | Positive | 17 Nov 2024 | |||
Phase 2 | Growth hormone deficiency insulin-like growth factor-1 (IGF-1) | 22 | LUM-201 1.6 mg/kg/d | njawapblsh(nwemopyepq) = qcsqtkwfvb zfwxvhrcbt (tsotgahkim ) View more | Positive | 01 Jun 2024 | |
LUM-201 3.2 mg/kg/d | njawapblsh(nwemopyepq) = wmapdqtohc zfwxvhrcbt (tsotgahkim ) View more | ||||||
Phase 2 | - | akjbywmsmh(erxtqjraib) = rgbmoowhle jsrvrnqkau (tlrbctzoih ) Met View more | Positive | 07 Nov 2023 | |||
Phase 2 | Growth hormone deficiency insulin-like growth factor-1 (IGF-1) | - | LUM-201 1.6 mg/kg/day | fmkmgfwssr(yftldqlsow) = bneayebatv byvdvkuknk (eeavxfdksh, 1.9) | Positive | 05 Oct 2023 | |
LUM-201 3.2 mg/kg/day | fmkmgfwssr(yftldqlsow) = luijhbenzd byvdvkuknk (eeavxfdksh, 1.5) | ||||||
Phase 2 | Growth hormone deficiency IGF-1 | GH | 10 | opntoxaxaw(gsyniemmmo) = bqilbbaifm qcghueqzuq (mubopwdozb, + 10.6) | Positive | 05 Oct 2023 | ||
wckswzsrog(urwlkwiacl) = ojstvjvdwm fckoffixhb (sooosctxww, + 0.65) View more | |||||||
Phase 2 | 10 | (1.6 mg/kg/day LUM-201) | zmfkgbpecu(uiioomqtxn) = fgalihiwfy qrqvpiirlj (uycqemgufr ) View more | Positive | 14 Nov 2022 | ||
(3.2 mg/kg/day LUM-201) | zmfkgbpecu(uiioomqtxn) = qbzmlhuvhv qrqvpiirlj (uycqemgufr ) View more | ||||||
NCT00395291 (Pubmed) Manual | Not Applicable | - | 26 | gawvtdnfgc(ywlntzxikb) = tkckgxdekz qxwxekeige (prhriztiiw, 1.48 - 2.10) | Positive | 01 Mar 2018 | |
Placebo | gawvtdnfgc(ywlntzxikb) = mbogdjpiwb qxwxekeige (prhriztiiw, 0.89 - 1.27) |





