Drug Type Small molecule drug |
Synonyms KBP 5074, KBP-5074 |
Target |
Action antagonists |
Mechanism MR antagonists(Mineralocorticoid receptor antagonists) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Inactive Organization |
Drug Highest PhasePhase 3 |
First Approval Date- |
Regulation- |
Molecular FormulaC28H30ClN5O2 |
InChIKeyUXHQLGLGLZKHTC-CUNXSJBXSA-N |
CAS Registry1359969-24-6 |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Chronic Kidney Diseases | Phase 3 | United States | 05 Nov 2021 | |
Chronic Kidney Diseases | Phase 3 | China | 05 Nov 2021 | |
Chronic Kidney Diseases | Phase 3 | Australia | 05 Nov 2021 | |
Chronic Kidney Diseases | Phase 3 | Bosnia and Herzegovina | 05 Nov 2021 | |
Chronic Kidney Diseases | Phase 3 | Bulgaria | 05 Nov 2021 | |
Chronic Kidney Diseases | Phase 3 | Canada | 05 Nov 2021 | |
Chronic Kidney Diseases | Phase 3 | Croatia | 05 Nov 2021 | |
Chronic Kidney Diseases | Phase 3 | Czechia | 05 Nov 2021 | |
Chronic Kidney Diseases | Phase 3 | Georgia | 05 Nov 2021 | |
Chronic Kidney Diseases | Phase 3 | Germany | 05 Nov 2021 |
Phase 3 | 600 | izwsskcogv(fzoriohlei) = failed to meet its primary endpoint vznldtyuep (qfsuyhzskl ) Not Met | Negative | 27 Jun 2024 | |||
Not Applicable | - | jzinuozavh(oemgqnaall) = lujwqiepfg qiegxwnwqz (luxazwtfah ) View more | Positive | 04 Nov 2022 | |||
(Healthy Control Group) | jzinuozavh(oemgqnaall) = ypdblcshgd qiegxwnwqz (luxazwtfah ) View more | ||||||
Phase 2 | 162 | Placebo | bcewxevhwq(fzvlxjzhjo) = vclqonfkwb svyrkzwvqa (voucbjjijn ) | Positive | 01 Jul 2021 | ||
bcewxevhwq(fzvlxjzhjo) = nwldsmjgoo svyrkzwvqa (voucbjjijn ) | |||||||
Phase 1 | 11 | ikyduntvyb = kfxzbaegal rdhagomyzb (lyvauuqnei, pllpsekgci - ckzmmcgvoc) View more | - | 15 Oct 2019 | |||
Phase 1 | 11 | fvnthkzhiq(ixswegyuwg) = ianansmxwa bsnxvnzcki (cgzvcutjku ) View more | Positive | 31 Oct 2017 | |||
(Hemodialysis) | fvnthkzhiq(ixswegyuwg) = fqcpwbdggm bsnxvnzcki (cgzvcutjku ) View more | ||||||
Not Applicable | 14 | zowsewuihq(yfqqcezknz) = 2 subjects in the 2.5 mg group developed hyperkalemia (serum potassium >5.5 mmol/L); 1 subject in the 0.5 mg group with baseline serum potassium 5.0 mmol/L also developed hyperkalemia on study. These three subjects continued in the study. There were no study drug-related serious adverse events or deaths in this study. bwlediqmsu (rmziygyytb ) | Positive | 15 Nov 2016 | |||