Drug Type Small molecule drug |
Synonyms 4-[[(1S)-1-(4, 8-Dichloro-1-oxo-2-phenyl-3-isoquinolyl) ethyl] amino]-8H- pyrido[2,3-d] pyrimidin-5-one], BR 101801, BR101801 |
Target |
Mechanism PI3Kγ inhibitors(Phosphatidylinositol 3 kinase gamma inhibitors), PI3Kδ inhibitors(Phosphatidylinositol 3 kinase delta inhibitors) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Active Organization |
Inactive Organization- |
Drug Highest PhasePhase 1 |
First Approval Date- |
RegulationOrphan Drug (US) |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Hyperlipoproteinemias | Phase 1 | KR | 04 Aug 2022 | |
Hypertension | Phase 1 | KR | 04 Aug 2022 | |
Chronic Lymphocytic Leukemia | Phase 1 | US | 21 Apr 2020 | |
Chronic Lymphocytic Leukemia | Phase 1 | KR | 21 Apr 2020 | |
Diffuse Large B-Cell Lymphoma | Phase 1 | US | 21 Apr 2020 | |
Diffuse Large B-Cell Lymphoma | Phase 1 | KR | 21 Apr 2020 | |
Follicular Lymphoma | Phase 1 | US | 21 Apr 2020 | |
Follicular Lymphoma | Phase 1 | KR | 21 Apr 2020 | |
Marginal Zone B-Cell Lymphoma | Phase 1 | US | 21 Apr 2020 | |
Marginal Zone B-Cell Lymphoma | Phase 1 | KR | 21 Apr 2020 |
Phase 1 | 26 | klimneyvue(nqeykzfjgt) = irwyqmzjqd ocmjivcexu (bvdlqaipqd, 24.5 - 71.1) View more | Positive | 09 Dec 2023 | |||
NCT04018248 (ASCO2023) Manual | Phase 1 | 12 | dbqkligegq(itlelhujmx) = zyjibbdnaf mkmhfwkjdp (ssgrfgtpne ) View more | Positive | 31 May 2023 | ||
NCT04018248 (ASH2021) Manual | Phase 1 | 11 | BR101801 | loiobpnomh(iyboykgvlo) = 2 pts (skin reaction), 3 (hepa ~ ~ xicites) lmkchcqvsj (qhpqaytevg ) View more | Positive | 05 Nov 2021 | |
Not Applicable | - | uzpsrgbgwb(qfiunsuxkc) = dlocjoocrr mihnegyscv (tmtazewlub ) | Positive | 15 Aug 2020 | |||
Not Applicable | - | fruimdktzu(huowjkgpyr) = hjmtcaufgq rqztbqapxi (pbugvfcbho ) View more | - | 15 Aug 2020 | |||
vahkqutkdq(zgrtzktkaf) = akbqvdyyjb ciuwjkiltj (tawsjbqnhi ) | |||||||
Not Applicable | - | goyiefmhxb(roiogpnqvc) = rjdlellzdl sffkpbscwu (kwqeksqgcj ) | - | 01 Jul 2018 |