Last update 23 Jan 2025

Ibrilatazar

Overview

Basic Info

Drug Type
Small molecule drug
Synonyms
Sodium 2-hydroxylinoleate
+ [2]
Target
Mechanism
PPARα/γ agonists(PPAR alpha/gamma agonists)
Originator Organization
Drug Highest PhasePhase 2
First Approval Date-
RegulationSpecial Review Project (CN), Orphan Drug (EU)
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Structure/Sequence

Molecular FormulaC18H32O3
InChIKeyAFDSETGKYZMEEA-HZJYTTRNSA-N
CAS Registry57818-44-7

External Link

KEGGWikiATCDrug Bank
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R&D Status

10 top R&D records.
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IndicationHighest PhaseCountry/LocationOrganizationDate
NeuroblastomaPhase 2
ES
18 Jul 2023
Pancreatic CancerPhase 2
EU
30 Jan 2022
Pancreatic CancerPhase 2
EU
30 Jan 2022
Metastatic Pancreatic CancerPhase 2
ES
26 Apr 2021
Endometrial CarcinomaPhase 2
ES
-
Lung CancerPhase 2
ES
-
Squamous Cell CarcinomaDiscovery
CN
29 Oct 2018
Squamous non-small cell lung cancerDiscovery
ES
01 Dec 2016
Advanced cancerDiscovery
ES
01 Feb 2014
Advanced Malignant Solid NeoplasmDiscovery
ES
01 Feb 2014
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Clinical Result

Indication
Phase
Evaluation
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Study
Phase
PopulationAnalyzed EnrollmentGroupResultsEvaluationPublication Date
Phase 1/2
51
Ibrilatazar (ABTL0812) + Carboplatin/Paclitaxel
(The phase 1 part)
-
Positive
22 Jul 2024
Ibrilatazar (ABTL0812) + Carboplatin/Paclitaxel
(zljyvixsrf) = tmfqdlwpie izadfnnohz (dhwkoffcnq )
Phase 2
40
ABTL0812+Paclitaxel+Carboplatin
(ecuamplcbf) = uvswraizek ztrhvobfzv (wwleqkvdvw, 34.2 - 65.9)
Positive
26 May 2023
Not Applicable
22
(fuqdovjstb) = ascfugjitg spsbsxpmiy (ccwgsnpabp, 32.2 - 75.6)
-
29 Jan 2021
Phase 2
42
(smqdquhdxc) = tmcyiludea ebzftqsufi (svkzkmkmhv, 46 - 80)
Positive
17 Sep 2020
Phase 1
21
Paclitaxel+Carboplatin+ABTL 0812
(kbzattrqhd) = neutrophil count decreased (43%), nausea (24%), fatigue (19%), anemia, vomiting, dyspepsia, platelet count decreased, arthralgia and neurotoxicity (10% each) ykbvhrijfq (jssnruskpp )
Positive
01 Jun 2019
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Regulation

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