Last update 20 Mar 2025

Plazomicin Sulfate

Overview

Basic Info

Drug Type
Small molecule drug
Synonyms
Plazomicin, Plazomicin sulfate (USAN), [14C]-plazomicin
+ [2]
Action
inhibitors
Mechanism
30S subunit inhibitors(30S ribosomal subunit inhibitors), Protein biosynthesis inhibitors
Originator Organization
Active Organization
Drug Highest PhaseApproved
First Approval Date
United States (25 Jun 2018),
RegulationPriority Review (United States)
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Structure/Sequence

Molecular FormulaC25H48N6O10
InChIKeyIYDYFVUFSPQPPV-PEXOCOHZSA-N
CAS Registry1154757-24-0
View All Structures (2)

External Link

R&D Status

Approved
10 top approved records.
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IndicationCountry/LocationOrganizationDate
Pyelonephritis
United States
25 Jun 2018
Urinary Tract Infections
United States
25 Jun 2018
Developing
10 top R&D records.
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IndicationHighest PhaseCountry/LocationOrganizationDate
Kidney Failure, ChronicPhase 2
United States
05 Jan 2021
Gram-Negative Bacterial InfectionsPhase 2
China
31 Dec 2019
Acute pyelonephritisPhase 2-11 Jan 2016
Carbapenem Resistant Bacterial InfectionPhase 2-16 Sep 2014
Complicated urinary tract infectionPhase 2-16 Sep 2014
Hospital acquired bacterial pneumoniaPhase 2-16 Sep 2014
Pneumonia, Ventilator-AssociatedPhase 2-16 Sep 2014
SepsisPhase 2-16 Sep 2014
Renal InsufficiencyPhase 2-01 Sep 2011
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Clinical Result

Indication
Phase
Evaluation
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Study
Phase
PopulationAnalyzed EnrollmentGroupResultsEvaluationPublication Date
Phase 1
-
64
cujpzdcfcr(snzwwvyoqs) = udyntgitdr hkjwzitagx (vrexqumsel )
-
01 Nov 2019
Phase 3
609
(tgnyswprts) = odalmtqvjk tqqjwunhdm (qrtycdvzui )
Non-superior
21 Feb 2019
(tgnyswprts) = vkdfufrxeh tqqjwunhdm (qrtycdvzui )
Phase 3
69
(Plazomicin in Combination With Meropenem or Tigecycline)
pwnppejple(mhucihtltg) = rosnijrjwy rbnjndlbcp (ticsdfbkie, yhadsxnpvj - alebxmcene)
-
16 Oct 2018
(Colistin in Combination With Meropenem or Tigecycline)
pwnppejple(mhucihtltg) = cuqjqkzvuh rbnjndlbcp (ticsdfbkie, hhdpfoemoz - eaxuyrimaj)
Phase 3
609
bbrsqtgbkg(skfmcxikit) = jbgmvlxrjm jwofrzpysi (jrxgooyfhw, keoydsjysf - jaqjrhbabv)
-
23 Aug 2018
bbrsqtgbkg(skfmcxikit) = umvmzimjgg jwofrzpysi (jrxgooyfhw, diyhcsffha - kmsktyfkxv)
Phase 2
145
plazomicin+placebo
(Plazomicin (10 mg/kg))
mnwgqsqgjs(fmhpnjuenn) = utveqzikcm ltuvtlusjn (hrvgumgboa, ffyshxnzhm - htetqanryk)
-
22 Aug 2018
plazomicin+placebo
(Plazomicin (15 mg/kg))
mnwgqsqgjs(fmhpnjuenn) = dhxjonendn ltuvtlusjn (hrvgumgboa, eduxkpdqhm - urzsfkjruv)
Phase 2
145
wljosecvbz(uyuqqhlknk) = yxggptxnsn rccvdgnmai (xzxzjhmqch, 21.1 - 78.9)
-
01 Apr 2018
wljosecvbz(uyuqqhlknk) = cjadgnrmqr rccvdgnmai (xzxzjhmqch, 46.1 - 74.2)
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