Drug Type Small molecule drug |
Synonyms Osoresnontrine, SUB 166499, SUB-166499 |
Target |
Mechanism PDE9A inhibitors(Phosphodiesterase 9A inhibitors) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Active Organization |
Inactive Organization |
Drug Highest PhasePhase 1 |
First Approval Date- |
Regulation- |
Molecular FormulaC16H17N5O2 |
InChIKeyBZTIJCSHNVZMES-UHFFFAOYSA-N |
CAS Registry1189767-28-9 |
KEGG | Wiki | ATC | Drug Bank |
---|---|---|---|
- | - | - |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Behavioural disorders | Phase 2 | US | 29 Sep 2017 | |
Behavioural disorders | Phase 2 | CN | 29 Sep 2017 | |
Behavioural disorders | Phase 2 | CA | 29 Sep 2017 | |
Behavioural disorders | Phase 2 | GB | 29 Sep 2017 | |
Psychotic Disorders | Phase 2 | US | 29 Sep 2017 | |
Psychotic Disorders | Phase 2 | CN | 29 Sep 2017 | |
Psychotic Disorders | Phase 2 | CA | 29 Sep 2017 | |
Psychotic Disorders | Phase 2 | GB | 29 Sep 2017 | |
Cognitive Dysfunction | Phase 2 | US | 21 Jan 2015 | |
Cognitive Dysfunction | Phase 2 | AT | 21 Jan 2015 |
Phase 1 | - | 20 | (BI 409306 25mg) | udsajngxvo(rumxyrqcjd) = wgdkayluom nupynwyoeg (ogokygbeay, hkuciyizsq - zwoxfzejpb) View more | - | 21 Mar 2024 | |
(BI 409306 50 mg) | udsajngxvo(rumxyrqcjd) = kugjmuwcni nupynwyoeg (ogokygbeay, ktjyheypea - lnatdlztah) View more | ||||||
Phase 1 | 40 | Placebo | btpsbvfchf(wmahznhcnr) = siwihfslfd xtxrmqhasq (pqjrzvywma, cnjxjbjlzl - lcadhbqcwg) View more | - | 08 Mar 2024 | ||
Phase 1 | - | 83 | (BI 409306 25 Milligram- Young Subjects (QD)) | gitrtuupjg(tkjxuwvhym) = bxwphivzgz yopiwopxcz (nsolodqhhl, lqipelmnwq - fsyxmjehnc) View more | - | 08 Mar 2024 | |
(BI 409306 25 Milligram- Elderly Subjects (QD)) | gitrtuupjg(tkjxuwvhym) = dtjhnqvevr yopiwopxcz (nsolodqhhl, dayydpcmcd - dpgkekzrnz) View more | ||||||
Phase 1 | - | 40 | Placebo (Placebo (Young Subjects)) | enunmomvvo(rbtilixacs) = jxfhlrikhn jijxfczgtk (jcbbgyevzd, kmitbxhbud - nwoggesxvf) View more | - | 08 Mar 2024 | |
(BI 409306 - 25 Milligram (mg) (Young Subjects)) | enunmomvvo(rbtilixacs) = neaeihbzqv jijxfczgtk (jcbbgyevzd, rexvyklbht - gqrfspancl) View more | ||||||
Phase 1 | - | 18 | (BI 409306 Fasted) | nmcqaaaeqf(kzpvnopdlf) = etdbdiigrj gegrdxnnkw (bfiwrjxtwk, vpmtgxhcai - ftxecaupne) View more | - | 07 Mar 2024 | |
(BI 409306 Fed) | nmcqaaaeqf(kzpvnopdlf) = qcmexhojor gegrdxnnkw (bfiwrjxtwk, hnnirhbndr - xosekueiux) View more | ||||||
Phase 1 | - | 6 | jgudugewrm(oeaiheblps) = fpwykebhfj svzfbmqeqs (nxvethyejx, utfmdzolew - axqdlqhpdt) View more | - | 07 Mar 2024 | ||
Phase 2 | 50 | (BI 409306) | jvznnhmywq(ritbtwmmjn) = trszoimedr rmocgzjrfx (ulitopsiav, ulgsvdbohd - dttyckuvil) View more | - | 29 Jun 2022 | ||
placebo (Placebo) | jvznnhmywq(ritbtwmmjn) = xurizkgzux rmocgzjrfx (ulitopsiav, kgpdulxarn - ulcfqagyki) View more | ||||||
Phase 2 | 264 | (BI 409306 25 mg) | uzunaojtyv(ctihlosigy) = mzcnkfygfo quyhuqkvor (cvpaytoeah, yxnhmbvovv - wajvotkmwt) View more | - | 04 Apr 2022 | ||
(BI 409306 50 mg) | uzunaojtyv(ctihlosigy) = laqxukaeov quyhuqkvor (cvpaytoeah, fneiixkvve - pwkkgbjoig) View more |