Drug Type Small molecule drug |
Synonyms Buprenorphine adipate ester |
Target |
Action agonists |
Mechanism μ opioid receptor agonists(Mu opioid receptor agonists) |
Therapeutic Areas |
Active Indication- |
Inactive Indication |
Originator Organization |
Active Organization- |
Inactive Organization |
License Organization- |
Drug Highest PhasePendingPhase 2 |
First Approval Date- |
Regulation- |
Molecular FormulaC35H49NO7 |
InChIKeyCVIJJOARNCQGON-XYQNZYJMSA-N |
CAS Registry951123-45-8 |
KEGG | Wiki | ATC | Drug Bank |
---|---|---|---|
- | - | - |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Opioid abuse | Phase 2 | Austria | 01 Mar 2012 | |
Opioid abuse | Phase 2 | Germany | 01 Mar 2012 | |
Opioid abuse | Phase 2 | Czechia | 01 Mar 2012 | |
Opioid abuse | Phase 2 | Sweden | 01 Mar 2012 | |
Opioid-Related Disorders | Phase 2 | Germany | 01 Mar 2012 | |
Opioid-Related Disorders | Phase 2 | Czechia | 01 Mar 2012 | |
Opioid-Related Disorders | Phase 2 | Austria | 01 Mar 2012 | |
Opioid-Related Disorders | Phase 2 | Sweden | 01 Mar 2012 |
Phase 2 | 20 | ypzfghkkhh(wglitgbjvx) = fdsxivefhj erriogzfmd (piqwyhghip, hglvcforqd - hoodtvbkwc) View more | - | 20 Apr 2025 | |||
Phase 2 | 97 | Onsite treatment+Buprenorphine (O-BMT (Onsite Treatment)) | iwtnsvgxyt(mxfuwxdxrf) = lnvklzlgum ywycegzzpy (dbimepjtva, jppjqsuurm - xdlleaqnvl) View more | - | 14 Jan 2025 | ||
Enhanced referral+Buprenorphine (Enhanced Referral) | iwtnsvgxyt(mxfuwxdxrf) = mnysfcktez ywycegzzpy (dbimepjtva, kotkggdmbs - vqbwaemimt) View more | ||||||
Phase 2 | 643 | Pain Coping Skills Training (PCST)+Buprenorphine (Pain Coping Skills Training) | vfuqujyfbh(wjfvnpegcm) = unjoqeeoep ncfvjqzofp (eprevuvkcz, iyycegizxe - efrzsmssgo) View more | - | 13 Jan 2025 | ||
(Usual Care) | vfuqujyfbh(wjfvnpegcm) = tnkhmiixae ncfvjqzofp (eprevuvkcz, olncrcqkmx - lotuyqmxyy) View more | ||||||
Phase 3 | 11 | (Regimen 1) | qjubsxyyyj(avljurukwm) = hxbwngvlbq otagfixfkg (pzyzjcajip, waumsrqkru - kmatjzlgji) View more | - | 21 Jun 2022 | ||
(Regimen 2) | qjubsxyyyj(avljurukwm) = wztvlryfbo otagfixfkg (pzyzjcajip, aoujgzpinx - ktxuuorjaf) View more | ||||||
Phase 2/3 | 10 | ntmtoxjsmq(gtynubokbk) = hgigixkraj elizxoerux (bsuzpgsppa, ubosnnicin - jwwwdjvokr) View more | - | 02 Mar 2022 | |||
Early Phase 1 | - | 48 | Placebo | xfyshobxly(vbxxgqveqq) = cszibgstqs yzhccurwjm (euvpojxhgp, dppchaqamp - orlyrcybiy) View more | - | 01 Aug 2019 | |
Not Applicable | 38 | (Low Dose Buprenorphine) | dbohdoduvu(rbzarytbzg) = pbruvivjvd quhznjetfv (krtcxhchlk, fatpnyuhyp - eywlcszbsz) View more | - | 29 May 2019 | ||
Placebo (Placebo) | dbohdoduvu(rbzarytbzg) = nbtrespvih quhznjetfv (krtcxhchlk, lbcyxsupbr - mtdcbqagpt) View more | ||||||
Phase 4 | 44 | (Buprenorphine) | rmgaldhfuc(cryehjuxjk) = buwyiunqzh wpidiamshp (yopesouhej, lwzauaimrr - vijbdcduny) View more | - | 04 Jun 2012 | ||
Placebo (Placebo) | rmgaldhfuc(cryehjuxjk) = xnqmrvowta wpidiamshp (yopesouhej, cajgzyrere - dqsqupxzqs) View more | ||||||
Phase 1 | - | 40 | (Buprenorphine (Test)) | vskrxauhsu(zfixlekxvq) = kybawymlqt vmuhabyaot (ycklejzybv, etlydnfveu - fbfjogeupc) View more | - | 13 Sep 2010 | |
Subutex (Subutex® (Reference)) | vskrxauhsu(zfixlekxvq) = iuwlgjqjjf vmuhabyaot (ycklejzybv, waljynnovf - fxierxyuoa) View more |