Drug Type Small molecule drug |
Synonyms ATZ/RTV |
Target |
Action inhibitors |
Mechanism HIV-1 pol inhibitors(Human immunodeficiency virus type 1 Pol protein inhibitors) |
Therapeutic Areas |
Active Indication |
Inactive Indication- |
Originator Organization |
Active Organization |
Inactive Organization |
License Organization- |
Drug Highest PhaseNDA/BLA |
First Approval Date- |
Regulation- |
Molecular FormulaC38H54N6O11S |
InChIKeyDQSGVVGOPRWTKI-QVFAWCHISA-N |
CAS Registry229975-97-7 |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
HIV Infections | NDA/BLA | United States | - | |
HIV Infections | NDA/BLA | United States | - |
Phase 4 | 1 | (Efavirenz 600 mg) | ftlgmmrapw(isbsackxgf) = jwacllvbrk xheltglkuh (ltqkoyvxyy, wykduecoft - dtshjmyepz) View more | - | 11 Aug 2017 | ||
(Arm B - Atazanavir/Ritonavir) | ftlgmmrapw(isbsackxgf) = ezqrmuhvdr xheltglkuh (ltqkoyvxyy, ldbrzigogn - impvluspfe) View more | ||||||
Phase 3 | 286 | ommznlosgm(ptvxpimpms) = drtoycfbff pjzqtqwsuy (gbdbgyiuqf ) View more | Non-inferior | 01 Jan 2017 | |||
2NUCs+Atazanavir/Ritonavir | ommznlosgm(ptvxpimpms) = rxqinckmqc pjzqtqwsuy (gbdbgyiuqf ) View more | ||||||
Not Applicable | 10 | rpeahsttol(ydztuatirv) = dnazwtgcqd kmkvlirjkp (intundoujp ) | Positive | 01 Jan 2017 | |||
Phase 4 | 286 | Dual treatment with atazanavir-ritonavir plus lamivudine | wciauxlmve(prvhbswnwy) = lirsnhltns igitxhkeuj (jxsqeultkc ) | Positive | 01 Jul 2015 | ||
Triple treatment with atazanavir-ritonavir plus two nucleos(t)ides | wciauxlmve(prvhbswnwy) = nwqftvgmjw igitxhkeuj (jxsqeultkc ) | ||||||
Phase 4 | 108 | lkdanknpjp(unktqagcsj) = lxztdjlkgc akhnynlpxw (hspdbohfuv, 129 - 349) View more | - | 01 Jun 2015 | |||
Atazanavir/Ritonavir | lkdanknpjp(unktqagcsj) = qmfzawiyso akhnynlpxw (hspdbohfuv, 146 - 238) View more | ||||||
Not Applicable | HIV Infections Second line | 559 | irruilwexm(oeorwrpbot) = lfaonhtkvt koptigwxjo (atfdqmfsgh ) View more | Positive | 01 Jan 2015 | ||
irruilwexm(oeorwrpbot) = oqbtagrxzs koptigwxjo (atfdqmfsgh ) View more | |||||||
Not Applicable | 18 | Atazanavir/ritonavir 200/100 mg | duogpamirq(olueqlmuzc) = xyoijstskx hrbduknror (zsuflmeeqp ) | - | 01 Dec 2014 | ||
Phase 4 | 180 | Atazanavir/ritonavir | vgabkbrrnw(mlqtzlirgl) = xchqhnioqn bsvnfeonfh (inbctadxou ) View more | - | 01 Jul 2014 | ||
vgabkbrrnw(mlqtzlirgl) = jhroeqhwzw bsvnfeonfh (inbctadxou ) | |||||||
Not Applicable | First line | 2,167 | ttqlslpowe(ujbaesbaoa) = pbgwiuzwyb xgnqvjqlhs (pddtsiqzix ) View more | - | 01 Jan 2013 | ||
ttqlslpowe(ujbaesbaoa) = hpabvcjtll xgnqvjqlhs (pddtsiqzix ) View more | |||||||
Phase 4 | 219 | ATV+RTV (ATV/RTV Switch Arm) | wwlzeidhqz(dehjodgovp) = nfrkutupzo ixcvvgwbup (vnxngllcwj, 0.027) View more | - | 07 May 2010 | ||
PI+RTV (PI/RTV Control Arm) | wwlzeidhqz(dehjodgovp) = zxzcbrwefv ixcvvgwbup (vnxngllcwj, 0.036) View more |