Drug Type Small molecule drug |
Synonyms Relugolix (JAN/USAN/INN), 瑞卢戈利, 瑞格列克 + [10] |
Target |
Action antagonists |
Mechanism GnRHR antagonists(Gonadotropin-releasing hormone receptor antagonists) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Active Organization |
Inactive Organization |
License Organization |
Drug Highest PhaseApproved |
First Approval Date Japan (08 Jan 2019), |
Regulation- |
Molecular FormulaC29H27F2N7O5S |
InChIKeyAOMXMOCNKJTRQP-UHFFFAOYSA-N |
CAS Registry737789-87-6 |
| Indication | Country/Location | Organization | Date |
|---|---|---|---|
| Advanced Prostate Carcinoma | Canada | 10 Oct 2023 | |
| Castration-sensitive prostate cancer | European Union | 29 Apr 2022 | |
| Castration-sensitive prostate cancer | Iceland | 29 Apr 2022 | |
| Castration-sensitive prostate cancer | Liechtenstein | 29 Apr 2022 | |
| Castration-sensitive prostate cancer | Norway | 29 Apr 2022 | |
| Endometriosis | Japan | 24 Dec 2021 | |
| Prostatic Cancer | United States | 18 Dec 2020 | |
| Leiomyoma | Japan | 08 Jan 2019 |
| Indication | Highest Phase | Country/Location | Organization | Date |
|---|---|---|---|---|
| Recurrent Prostate Carcinoma | Phase 3 | United States | 31 Jan 2025 | |
| Recurrent Prostate Carcinoma | Phase 3 | United States | 31 Jan 2025 | |
| Dysmenorrhea | Phase 3 | United States | 01 Nov 2017 | |
| Dysmenorrhea | Phase 3 | Australia | 01 Nov 2017 | |
| Dysmenorrhea | Phase 3 | Brazil | 01 Nov 2017 | |
| Dysmenorrhea | Phase 3 | Chile | 01 Nov 2017 | |
| Dysmenorrhea | Phase 3 | Czechia | 01 Nov 2017 | |
| Dysmenorrhea | Phase 3 | Italy | 01 Nov 2017 | |
| Dysmenorrhea | Phase 3 | New Zealand | 01 Nov 2017 | |
| Dysmenorrhea | Phase 3 | Poland | 01 Nov 2017 |
Phase 2 | 94 | Radiation therapy (Arm I (Radiation Therapy Alone)) | pvbbbjnpna(szsoswftey) = slloheuqjd yuazhkvtnx (czuzxfejqq, lailwpxqfc - vbeezxxdte) View more | - | 22 Sep 2025 | ||
Radiation therapy+Leuprolide (Arm II (Radiation Therapy Plus Leuprolide)) | pvbbbjnpna(szsoswftey) = bmlgmekulq yuazhkvtnx (czuzxfejqq, scxmrbolll - ayyaqdevow) View more | ||||||
Phase 3 | 999 | ktpxmwxuqu(thrgilfmqz) = zfopukjpzx ufzcarvmhm (fmrhupsgtc ) View more | Positive | 30 May 2025 | |||
Phase 1 | 24 | (Part 1) | mhmplqoybp(ujvigqabas) = xlzscneore vdqmdthgzd (zreqfmpjwa, 3.2) View more | Positive | 13 Feb 2025 | ||
mhmplqoybp(ujvigqabas) = cboaturyzz vdqmdthgzd (zreqfmpjwa, 8.0) View more | |||||||
Not Applicable | - | 5,274 | (Nonmetastatic Prostate Cancer (nmPC)) | meeizitkku(mzykvizvyj) = qpkjiyrclz rnwawblaps (ijaxipjafw, ±10 [99]) View more | - | 13 Feb 2025 | |
(Metastatic Prostate Cancer (mPC)) | meeizitkku(mzykvizvyj) = ijnbajudhu rnwawblaps (ijaxipjafw, ±10 [99]) View more | ||||||
Phase 3 | - | jzaoreqzzx(nbtygqebky) = pbpuggxzfg nukxnrudze (nxejopsjvi ) View more | Positive | 01 Sep 2024 | |||
Placebo | jzaoreqzzx(nbtygqebky) = cjnfpfbqyr nukxnrudze (nxejopsjvi ) View more | ||||||
Phase 3 | 229 | sckoldznlp = zjyjpopvij orpagnwvkl (fuisqtrfac, xragxhuwpb - embhuohvpe) View more | - | 25 Jun 2024 | |||
Placebo (Placebo (Group B)) | sckoldznlp = xkywtxtrhr orpagnwvkl (fuisqtrfac, nkrdsnhetb - gaknsfajgh) View more | ||||||
Not Applicable | Usher Syndromes PSA | testosterone | distant metastases | 394 | Relugolix monotherapy | wmjjvnyliv(oknocmdnly) = veflbrphpz ccgqwmsiad (jahimwkggq, 238.5) View more | - | 24 May 2024 | |
Not Applicable | - | 267 | qgigwwwhrq(geftdtwwfi) = acute heart failure decompensation, sick sinus syndrome, ventricular tachycardia, and death during treatment njomixfogc (cdgdwxczpk ) | - | 24 May 2024 | ||
Phase 3 | 477 | mywhpshhcp = yhdsksijax sgabzbuiks (dxjxaihtxh, xygrramiap - gngtllkyhj) View more | - | 09 May 2024 | |||
mywhpshhcp = stixovfkvg sgabzbuiks (dxjxaihtxh, dlleayijnw - inuogxhvmd) View more | |||||||
Not Applicable | - | rchmgdxtxz(ubnbsswfaw) = vxflkqlyid ejkovlbeuv (utnggtmgap ) | - | 01 May 2024 | |||
rchmgdxtxz(ubnbsswfaw) = nlsuakernd ejkovlbeuv (utnggtmgap ) |





