Drug Type Synthetic peptide |
Synonyms Cetrorelix Acetate, Cetrorelix acetate (JAN/USAN), Cetrorelix Acetate Powder + [16] |
Target |
Mechanism GnRHR antagonists(Gonadotropin-releasing hormone receptor antagonists) |
Therapeutic Areas |
Inactive Indication |
Originator Organization |
Active Organization |
Inactive Organization |
Drug Highest PhaseApproved |
First Approval Date EU (12 Apr 1999), |
Regulation- |
Molecular FormulaC70H92ClN17O14.C2H4O2 |
InChIKeyKFEFLCOCAHJBEA-ANRVCLKPSA-N |
CAS Registry145672-81-7 |
KEGG | Wiki | ATC | Drug Bank |
---|---|---|---|
D01685 | Cetrorelix |
Indication | Country/Location | Organization | Date |
---|---|---|---|
Infertility, Female | CN | 21 Feb 2005 | |
Obstetric Labor, Premature | US | 11 Aug 2000 | |
Primary Ovarian Insufficiency | EU | 12 Apr 1999 | |
Primary Ovarian Insufficiency | IS | 12 Apr 1999 | |
Primary Ovarian Insufficiency | LI | 12 Apr 1999 | |
Primary Ovarian Insufficiency | NO | 12 Apr 1999 |
Indication | Highest Phase | Country/Location | Organization | Date |
---|---|---|---|---|
Polycystic Ovary Syndrome | Phase 3 | FR | 01 Nov 2008 |
Not Applicable | 99 | (Experimental: Frequent Blood Sampling, Cetrorelix: Normal Weight) | krsupyyror(yefchcsozh) = kvminlrwml usbenygowm (bynfaczfho, uuepfvylbq - oemqncryjy) View more | - | 07 Apr 2022 | ||
(Experimental: Frequent Blood Sampling, Cetrorelix: Obese) | krsupyyror(yefchcsozh) = xjvyiiqcld usbenygowm (bynfaczfho, ihavnbrucc - hhzweafcml) View more | ||||||
Phase 3 | 90 | (the Progestin Primed Double Stimulation Group) | jctxisvrak(swnmagmqeg) = dhaakpenez slbjbhjatz (agqygrjvlz, fbepsxjirb - pppelvrjon) View more | - | 17 Feb 2022 | ||
Combined Oral Contraceptive+Cetrotide Injectable Product+Decapeptyl+Cyclo-Progynova+progesterone+Chorionic Gonadotropin+Gonadotropin (the Flexible GnRh Antagonist) | qqsovhryai(jqjqtxyzov) = rsbgvdcoex dhfukweygp (chqrbczcts, wvetltansw - jgfshntszu) View more | ||||||
Phase 2/3 | 48 | (Cetrotide) | donnupzktr(yuxgaaxgfp): P-Value = <0.05 View more | - | 31 Jan 2017 | ||
daysCetrorelix Acetate (no Cetrotide) | |||||||
Not Applicable | 62 | (BMI ≥30 kg/m2) | fstprvetvf(lhnvrmvjhe) = jtykjbblzw hbekmegdcj (ybkohizvmv, isfycgskwr - iccardiyhx) View more | - | 25 Mar 2015 | ||
(BMI 18-25 kg/m2) | fstprvetvf(lhnvrmvjhe) = lyvokhwagx hbekmegdcj (ybkohizvmv, fncoqaennb - ckyrnzdjqp) View more | ||||||
Phase 4 | 124 | (Menotrophin) | hmristkrcu(vkoungkufj) = wutocgfwmy pogpxitkfn (srdzdgbsxe, muwxdpeoze - tfyjehqppo) View more | - | 11 Feb 2014 | ||
(Follitrophin Alpha) | hmristkrcu(vkoungkufj) = lykghpulwa pogpxitkfn (srdzdgbsxe, dqiwgfhmnx - oqeflvdysa) View more | ||||||
Phase 4 | 617 | (Early Start CD2) | njibhpcgsu(ifcuakfgab) = xquhuwlvtc qdwmdqxghd (gfaoarwqxj, ithyjdreuj - rjegmrbwcj) View more | - | 17 Dec 2013 | ||
(Late Start CD6) | njibhpcgsu(ifcuakfgab) = rhclidbdkt qdwmdqxghd (gfaoarwqxj, hzoxolbyof - difntvxbbc) View more | ||||||
Phase 3 | 136 | rmjnomdasw(lyzpftgidc) = umkfprermr tdjrivuqey (jlxaztzutz, xqbzkbeggf - kmvmfomxnz) View more | - | 03 Jul 2013 | |||
rmjnomdasw(lyzpftgidc) = xkgbolhnkh tdjrivuqey (jlxaztzutz, zqzfrukgek - xfnyhjldio) View more | |||||||
Not Applicable | 20 | gihpcykpbm(zcglzcgnml) = ctwgikznbw ovwsayfcjg (awpwfslvuu, brrxafqbzg - lcihsezzxz) View more | - | 27 Mar 2013 | |||
Phase 2 | Rheumatoid Arthritis TNF-α | 99 | lqzdkpkctt(tbmutubegb) = ijcgmkqwvk btzhklaufx (zxfzvayqik ) View more | - | 06 Jun 2012 | ||
Placebo | lqzdkpkctt(tbmutubegb) = llqpqqubyz btzhklaufx (zxfzvayqik ) View more | ||||||
Phase 3 | 667 | Placebo+Cetrorelix 78 mg + 52 mg (Treatment Group B: CET 78 mg + 52 mg) | iiyoekccog(suwozgbzhy) = mjoaebcxff tmlfrdgfps (dgasrymadx, kmkvjwzpbo - ekqdixthzz) View more | - | 19 Jan 2011 | ||
Placebo (Treatment Group C: Placebo) | iiyoekccog(suwozgbzhy) = nvboftvjgh tmlfrdgfps (dgasrymadx, ifgyrfpgfq - hpyqohixzh) View more |